SCHEMBL8784394

SCHEMBL8784394

COc1nc2cc(Cl)c(Cl)c(CCCl)c2nc1OC

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.35
PTGES O14684 1/20 0.33
NQO2 P16083 1/20 0.33
PGK1 P00558 2/20 0.32
GSK3B P49841 1/20 0.32
MAP4K2 Q12851 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784365 0.88 HRH4 (0.34) HRH4PTGESNQO2PGK1GSK3B
SCHEMBL8784616 0.85 TLR8 (0.35) HRH4PTGESNQO2PGK1
SCHEMBL7466499 0.84 HRH4 (0.35) HRH4PTGESNQO2PGK1GSK3B
SCHEMBL7468650 0.82 HRH4 (0.34) HRH4PTGESNQO2PGK1GSK3B
SCHEMBL8647402 0.82 PTGES (0.30) HRH4PTGES
SCHEMBL7825014 0.81 HDAC1 (0.31)
SCHEMBL7467268 0.80 GLP1R (0.34) HRH4PTGESNQO2
SCHEMBL8783998 0.79 CD274 (0.39)
SCHEMBL7470559 0.79 HRH4 (0.32) HRH4PTGESPGK1GSK3BMAP4K2
SCHEMBL7473964 0.77 HRH4 (0.39) HRH4PTGESNQO2PGK1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781279-A1 QUINOXALINEDIONE NMDA RECEPTOR ANTAGONISTS Pfizer Limited (GB) 1997-07-02 EP disclosed