SCHEMBL7471440

SCHEMBL7471440

O=C(O)c1ccc2[nH]c(-c3ccc([N+](=O)[O-])s3)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 5/20 0.45
HDAC6 Q9UBN7 3/20 0.42
RAB9A P51151 4/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
NPC1 O15118 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NR4A2 P43354 1/20 0.40
KMT2A Q03164 1/20 0.40
HSP90AA1 P07900 1/20 0.39
ESR2 Q92731 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NPBWR1 P48145 1/20 0.39
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
CASP6 P55212 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467865 0.86 RHEB (0.45) HDAC6RAB9AKDM4EALDH1A1HPGD
SCHEMBL19223667 0.81 KDM4E (0.57) CHEK2HDAC6RAB9AKDM4EALDH1A1
SCHEMBL3863014 0.80 CSNK2A2 (0.49) CHEK2HDAC6RAB9AKDM4EALDH1A1
SCHEMBL7464927 0.80 CHEK2 (0.49) CHEK2RAB9AKDM4EALDH1A1HPGD
SCHEMBL7472954 0.80 CHEK2 (0.49) CHEK2RAB9AKDM4EALDH1A1HPGD
SCHEMBL7470449 0.80 MAPT (0.39) HDAC6RAB9AALDH1A1NPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL7466334 0.78 MAPT (0.38) HDAC6MAPT
SCHEMBL12713528 0.78 RAB9A (0.60) HDAC6RAB9AKDM4EALDH1A1HPGD
SCHEMBL18229582 0.78 HDAC6 (0.66) HDAC6
SCHEMBL828113 0.77 KDM4E (0.56) CHEK2RAB9AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711768-B1 BENZIMIDAZOLE DERIVATIVE MITSUI CHEMICALS INC (JP) 2002-02-13 EP disclosed
US-5852011-A Benzimidazole derivatives MITSUI CHEMICALS, INC. (JP) 1998-12-22 US disclosed
EP-0711768-A1 BENZIMIDAZOLE DERIVATIVE MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-05-15 EP disclosed