SCHEMBL7471677

SCHEMBL7471677

O=C1C(Cc2ccccc2)CS(=O)(=O)N1CS(=O)(=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
CMA1 P23946 1/20 0.37
MMP2 P08253 5/20 0.37
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MAOB P27338 1/20 0.36
FOLH1 Q04609 1/20 0.36
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
CRBN Q96SW2 2/20 0.35
DDB1 Q16531 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472990 0.80 HSD11B1 (0.41) HSD11B1ALDH1A1KMT2ANPC1RAB9A
SCHEMBL7472214 0.77 MMP2 (0.37) HSD11B1PSEN1PSEN2APH1BNCSTN
SCHEMBL7449485 0.76 HSD11B1 (0.38) HSD11B1ALDH1A1KMT2ANPC1RAB9A
SCHEMBL7476991 0.74 PSEN1 (0.35) HSD11B1PSEN1PSEN2APH1BNCSTN
SCHEMBL7469169 0.70 ROCK2 (0.36) HSD11B1CMA1ALDH1A1KMT2ANPC1
SCHEMBL7420571 0.63 CA12 (0.61) NPC1RAB9AGAA
Benzylsulfonylbenzene SCHEMBL780337 0.62 TSHR (0.68) MMP2ALDH1A1KMT2AMAPTTSHR
SCHEMBL22206479 0.62 BACE1 (0.46) ALDH1A1MAPT
SCHEMBL7441792 0.61 DDB1 (0.49) HSD11B1ALDH1A1KMT2ANPC1RAB9A
SCHEMBL28942364 0.61 HSD11B1 (0.59) HSD11B1ALDH1A1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739338-B1 SERINE PROTEASE INHIBITORS: DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE-1,1 DIOXIDE AND 3-OXO-1,2,5-THIADIAZOLIDINE-1,1-DIOXIDE UNIV WICHITA STATE (US) 2002-04-10 EP disclosed
US-5550139-A ANTIINFLAMMATORY AGENT, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT THE WICHITA STATE UNIVERSITY (US) 1996-08-27 US disclosed