SCHEMBL7472990

SCHEMBL7472990

O=C1C(Cc2ccccc2)CS(=O)(=O)N1CF

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.41
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MEN1 O00255 3/20 0.36
MAPT P10636 2/20 0.36
TSHR P16473 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471677 0.80 HSD11B1 (0.38) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7449485 0.80 HSD11B1 (0.38) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7469169 0.74 ROCK2 (0.36) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7476991 0.73 PSEN1 (0.35) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7473383 0.73 HSD11B1 (0.34) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7462751 0.70 GAA (0.41) ALDH1A1LMNACYP1A2CYP2C9CYP2C19
SCHEMBL7464643 0.69 GFER (0.41) KMT2ALMNACYP1A2CYP2C9CYP2C19
SCHEMBL7472214 0.68 MMP2 (0.37) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7434618 0.68 HSD11B1 (0.44) HSD11B1KMT2AALDH1A1NPC1RAB9A
SCHEMBL7465763 0.68 EP300 (0.44) KMT2AALDH1A1LMNACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739338-B1 SERINE PROTEASE INHIBITORS: DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE-1,1 DIOXIDE AND 3-OXO-1,2,5-THIADIAZOLIDINE-1,1-DIOXIDE UNIV WICHITA STATE (US) 2002-04-10 EP disclosed
US-5550139-A ANTIINFLAMMATORY AGENT, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT THE WICHITA STATE UNIVERSITY (US) 1996-08-27 US disclosed