SCHEMBL7472201

SCHEMBL7472201

CCOC(=O)c1[c]cccc1OC(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
CYP1A2 P05177 1/20 0.39
TSHR P16473 1/20 0.38
ACHE P22303 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
MAPT P10636 4/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7475976 0.85 SLC6A3 (0.35) CYP1A2TSHRCA12CA1CA2
SCHEMBL7476308 0.83 KDM4E (0.49) CYP1A2TSHRACHECA12CA1
SCHEMBL7474724 0.83 HSD17B2 (0.45) CYP1A2TSHRCA12CA1CA2
SCHEMBL7594026 0.75 ELANE (0.35)
SCHEMBL7481962 0.73 CA12 (0.58) CYP1A2TSHRCA12CA1CA2
SCHEMBL1452206 0.73 TSHR (0.61) CYP1A2TSHRCA12CA1CA2
SCHEMBL27749672 0.72 ALDH1A1 (0.56) CYP1A2TSHRCA12CA1CA2
SCHEMBL7474112 0.69 L3MBTL1 (0.37) CYP1A2TSHRKDM4EHSD17B10LMNA
SCHEMBL7182176 0.68 L3MBTL1 (0.43) TSHRMAPTHSD17B10NPSR1
SCHEMBL28404237 0.68 ELANE (0.47) HDAC6TSHRACHEMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194417-A1 PHENOXY FLUOROPYRIMIDINES BAYER AG (DE) 2002-04-10 EP claimed
WO-2000078733-A1 PHENOXY FLUOROPYRIMIDINES BAYER AKTIENGESELLSCHAFT (DE) 2000-12-28 WO claimed
EP-1194417-A1 PHENOXY FLUOROPYRIMIDINES BAYER AG (DE) 2002-04-10 EP disclosed
WO-2000078733-A1 PHENOXY FLUOROPYRIMIDINES BAYER AKTIENGESELLSCHAFT (DE) 2000-12-28 WO disclosed