SCHEMBL7472634

SCHEMBL7472634

O=C1C(CCO)Oc2ccc(F)cc2N1Cc1cccc([N+](=O)[O-])c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
TSHR P16473 2/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
IDO1 P14902 1/20 0.40
CASP1 P29466 2/20 0.38
CASP3 P42574 2/20 0.38
CASP7 P55210 2/20 0.38
CASP4 P49662 1/20 0.38
CASP9 P55211 1/20 0.38
CASP6 P55212 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472270 0.88 ALDH1A1 (0.55) ALDH1A1HPGDHTTTSHRUSP2
SCHEMBL7470312 0.87 ALDH1A1 (0.48) ALDH1A1HPGDHTTTSHRUSP2
SCHEMBL7478182 0.82 ALDH1A1 (0.44) ALDH1A1HPGDHTTTSHRUSP2
SCHEMBL7469541 0.80 KMT2A (0.57) ALDH1A1TSHRUSP2LMNAMAPK1
SCHEMBL7474357 0.80 CASP1 (0.53) ALDH1A1HPGDHTTTSHRLMNA
SCHEMBL7472359 0.80 CASP1 (0.43) ALDH1A1HPGDHTTTSHRUSP2
SCHEMBL189949 0.80 MAPT (0.44) ALDH1A1TSHRUSP2LMNAMAPK1
SCHEMBL7477205 0.79 KMT2A (0.67) ALDH1A1HTTTSHRUSP2LMNA
SCHEMBL8557110 0.78 ALDH1A1 (0.36) ALDH1A1HPGDTSHRUSP2LMNA
SCHEMBL7468750 0.77 CASP3 (0.44) ALDH1A1HPGDHTTTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869949-B1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO MCNEIL PHARM INC (US) 2002-12-18 EP disclosed
US-5854242-A Benzoxazine antimicrobial agents ORTHO PHARMACEUTICAL CORPORATION (US) 1998-12-29 US disclosed
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
US-5696117-A BACTERICIDE ORTHO PHARMACEUTICAL CORPORATION (US) 1997-12-09 US disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed