SCHEMBL7472775

SCHEMBL7472775

O=C(O)Cn1c(=O)n(S(=O)(=O)c2cccnc2)c(=O)c2ccc(Cl)cc21

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.44
AKR1A1 P14550 1/20 0.44
MCL1 Q07820 1/20 0.40
KMO O15229 1/20 0.39
GABRA5 P31644 2/20 0.39
GABRA1 P14867 1/20 0.39
PTGDR2 Q9Y5Y4 3/20 0.39
MAT2A P31153 2/20 0.38
PPARG P37231 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
HTT P42858 3/20 0.38
HDAC6 Q9UBN7 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
USP2 O75604 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470400 0.88 AKR1B1 (0.49) AKR1B1AKR1A1PTGDR2PPARGPPARD
SCHEMBL7468729 0.87 MAPT (0.46) SMN1; SMN2
SCHEMBL7461621 0.86 KDM4E (0.38) MCL1GABRA5GABRA1MAT2APPARG
SCHEMBL7465874 0.85 AKR1B1 (0.50) AKR1B1AKR1A1KMOPTGDR2PPARG
SCHEMBL7457276 0.84 MAPT (0.47) SMN1; SMN2NPSR1
SCHEMBL7471563 0.81 PPARG (0.48) AKR1B1AKR1A1MCL1PTGDR2PPARG
SCHEMBL7468043 0.81 MAPT (0.48) SMN1; SMN2
SCHEMBL7465813 0.80 ALDH1A1 (0.43) SMN1; SMN2NPSR1
Iodide SCHEMBL7466550 0.80 MAPT (0.38) MAT2ASMN1; SMN2
SCHEMBL8705100 0.79 HTT (0.38) MCL1MAT2AHTTSMN1; SMN2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed