SCHEMBL7473702

SCHEMBL7473702

COC(=O)Cc1cc(C)c(C(=O)c2ccc(OC)cc2)n1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.56
ABCB11 O95342 1/20 0.56
ALDH1A1 P00352 4/20 0.53
LMNA P02545 3/20 0.53
CYP1A2 P05177 1/20 0.53
TSHR P16473 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
AKR1C3 P42330 3/20 0.45
PKM P14618 1/20 0.42
ALOX15 P16050 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
AKR1C2 P52895 1/20 0.41
RAB9A P51151 2/20 0.40
NPC1 O15118 2/20 0.40
GAA P10253 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9030622 0.87 PTGS2 (0.74) PTGS2ABCB11ALDH1A1LMNACYP1A2
Perchlorate SCHEMBL10997108 0.81 AKR1C3 (0.39) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL7674536 0.78 PTGS2 (0.57) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL4601841 0.77 CXCL8 (0.55) PTGS2ALDH1A1LMNAALOX15NPSR1
SCHEMBL11810694 0.77 ABCB11 (0.51) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL11190775 0.77 ALDH1A1 (0.42) PTGS2ABCB11ALDH1A1LMNASMN1; SMN2
SCHEMBL11001456 0.76 ABCB11 (0.45) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL10904870 0.76 PTGS2 (0.65) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL7676885 0.76 PTGS2 (0.55) PTGS2ABCB11ALDH1A1LMNACYP1A2
SCHEMBL11500022 0.76 PTGS2 (0.69) PTGS2ABCB11ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906279-B1 PYRROLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-6136844-A ANTIINFLAMMATORY AGENT; AUTOIMMUNE DISEASE SYNTEX (U.S.A.) INC. (US) 2000-10-24 US disclosed
US-6127402-A AN INHIBITORS OF PROSTAGLANDIN G/H SYNTHASE AND ARE ANTI-INFLAMMATORY AND ANALGESIC AGENTS SYNTEX (U.S.A.) INC. (US) 2000-10-03 US disclosed
US-5952368-A AN INHIBITORS OF PROSTAGLANDIN G/H SYNTHASE, ANTIINFLAMMATORY AND ANALGESIC AGENTS SYNTEX (U.S.A.) INC. (US) 1999-09-14 US disclosed
EP-0906279-A1 NOVEL PYRROLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-04-07 EP disclosed
WO-1997046524-A1 NOVEL PYRROLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-12-11 WO disclosed