SCHEMBL7474277

SCHEMBL7474277

CC(=O)OCC(=O)c1ccc2c(c1)C(C)(C)CN2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 3/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP26A1 O43174 1/20 0.41
CYP26B1 Q9NR63 1/20 0.41
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
MAPT P10636 2/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11810345 0.80 RARB (0.44) RARARARBRARGMAPTL3MBTL1
SCHEMBL31456579 0.77 RARB (0.53) ALDH1A1KDM4ETP53HSD17B10CYP3A4
SCHEMBL5734170 0.68 HSPA9 (0.49) KDM4EMAPTSMN1; SMN2NPSR1L3MBTL1
SCHEMBL28286506 0.67 ESR1 (0.59) ALDH1A1KDM4EHPGDTP53HSD17B10
SCHEMBL11758571 0.67 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDTP53HSD17B10
SCHEMBL16494210 0.67 MRGPRX2 (0.41) RARARARBRARG
SCHEMBL11754844 0.66 ALDH1A1 (0.61) ALDH1A1KDM4EHPGDTP53HSD17B10
SCHEMBL4828375 0.66 NPC1 (0.70) ALDH1A1KDM4EHPGDTP53MAPT
SCHEMBL15677052 0.66 MAPT (0.38) ALDH1A1TP53MAPTSMN1; SMN2L3MBTL1
Hydrochloric Acid SCHEMBL16494285 0.66 MRGPRX2 (0.40) RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216239-A1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2002-06-26 EP disclosed
WO-2001023374-A1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2001-04-05 WO disclosed