SCHEMBL7474346

SCHEMBL7474346

COC(=O)c1c(C=O)c(C)c(C)n1CC(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 2/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480610 0.82 ALDH1A1 (0.31) RAB9AALDH1A1
SCHEMBL7480607 0.82 ALDH1A1 (0.31) RAB9AALDH1A1
SCHEMBL7479670 0.81 MEN1 (0.36) RAB9ACYP3A4MEN1KMT2AALDH1A1
SCHEMBL7477896 0.80 MEN1 (0.33) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL7487012 0.79 KDM4E (0.37) MEN1KMT2AALDH1A1
SCHEMBL7478235 0.79 ADORA2B (0.31) MEN1KMT2A
SCHEMBL7482378 0.78 ALDH1A1 (0.37) CYP3A4MEN1KMT2AALDH1A1LMNA
SCHEMBL7475018 0.78 KDM4E (0.32) RAB9ACYP3A4ALDH1A1LMNAMAPT
SCHEMBL7478519 0.77 ALDH1A1 (0.33) RAB9AALDH1A1LMNAMAPTNPSR1
SCHEMBL7478089 0.77 KDM4E (0.32) ALDH1A1LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed