SCHEMBL7480607

SCHEMBL7480607

COC(=O)c1c(C=O)c(C)c(C)n1C/C=C/C(F)(F)F

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480610 1.00 ALDH1A1 (0.31) ALDH1A1POLBRAB9A
SCHEMBL7478519 0.85 ALDH1A1 (0.33) ALDH1A1POLBRAB9A
SCHEMBL7478131 0.84 ALDH1A1 (0.32) ALDH1A1POLBRAB9A
SCHEMBL7478128 0.84 ALDH1A1 (0.32) ALDH1A1POLBRAB9A
SCHEMBL7482378 0.83 ALDH1A1 (0.37) ALDH1A1POLB
SCHEMBL7474346 0.82 NPC1 (0.32) ALDH1A1RAB9A
SCHEMBL7478235 0.81 ADORA2B (0.31)
SCHEMBL7483009 0.78 ALDH1A1 (0.34) ALDH1A1
SCHEMBL7479670 0.78 MEN1 (0.36) ALDH1A1POLBRAB9A
SCHEMBL7477197 0.78 MAPT (0.43) ALDH1A1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed