SCHEMBL7474495

SCHEMBL7474495

[c]1oc2cccc(-c3ccc4ccccc4n3)c2c1-c1nccc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.39
RAB9A P51151 6/20 0.36
NPC1 O15118 5/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
HCRTR1 O43613 1/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 1/20 0.36
PDE10A Q9Y233 3/20 0.34
TOP2A P11388 1/20 0.33
KDM4E B2RXH2 5/20 0.33
LMNA P02545 2/20 0.33
GAA P10253 1/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18274771 0.92 RAB9A (0.37) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL15573918 0.76 AR (0.38) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL7808907 0.75 KDM4E (0.42) RAB9ANPC1ALDH1A1MAPTKMT2A
SCHEMBL29610252 0.73 RAB9A (0.49) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL15775443 0.73 RAB9A (0.49) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL3835162 0.72 RAB9A (0.50) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL7471796 0.72 AR (0.36) ARRAB9ANPC1MAPTKMT2A
SCHEMBL15590910 0.71 NPC1 (0.53) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL29775064 0.71 NPC1 (0.53) ARRAB9ANPC1ALDH1A1MAPT
SCHEMBL240495 0.69 AR (0.55) ARRAB9ANPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244653-A1 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2002-10-02 EP claimed
WO-2001046176-A2 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-06-28 WO claimed
EP-1244653-A1 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2002-10-02 EP disclosed
WO-2001046176-A2 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-06-28 WO disclosed