SCHEMBL7475321

SCHEMBL7475321

CCN(CC)CCN1CC(=O)N=C(c2ccccn2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 6/20 0.36
HPGD P15428 2/20 0.36
HTR1A P08908 1/20 0.36
DRD3 P35462 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR3A P46098 1/20 0.36
KCNH2 Q12809 1/20 0.36
GHSR Q92847 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
CASP1 P29466 1/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
MITF O75030 1/20 0.35
POLB P06746 1/20 0.35
DNMT1 P26358 1/20 0.35
HTT P42858 1/20 0.35
RAD52 P43351 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diethylamine SCHEMBL7561727 0.81 CCKBR (0.35) CCKBRBRD4
SCHEMBL7478420 0.78 CCKBR (0.47) ALDH1A1CCKBR
SCHEMBL6304136 0.78 HTR1A (0.56) ACHEKDM4EALDH1A1HTR1ADRD3
SCHEMBL4992080 0.73 GABRP (0.44) KDM4EALDH1A1HPGDHTR1ADRD3
SCHEMBL6308282 0.67 GABRA1 (0.66) OPRK1KCNH2GHSRCCKBRBRD4
SCHEMBL7535136 0.66 CCKBR (0.42) CCKBRBRD4
SCHEMBL23479881 0.65 KMT2A (0.48) KDM4EALDH1A1HPGDL3MBTL1KMT2A
Hydrochloric Acid SCHEMBL31096518 0.65 KMT2A (0.47) KDM4EALDH1A1HPGDL3MBTL1KMT2A
Hydrochloric Acid SCHEMBL23202473 0.65 KMT2A (0.47) KDM4EALDH1A1HPGDL3MBTL1KMT2A
Diethylamine SCHEMBL6308096 0.63 CYP1A2 (0.51) KDM4EALDH1A1L3MBTL1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951466-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP claimed
WO-1998028268-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 1998-07-02 WO claimed
EP-0951466-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP disclosed
WO-1998028268-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 1998-07-02 WO disclosed