SCHEMBL7476769

SCHEMBL7476769

Cc1cccc(Nc2nccc(-c3cccnc3)n2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 15/20 1.00
BCR P11274 13/20 1.00
PRKCA P17252 11/20 0.73
SRC P12931 10/20 0.73
PRKCD Q05655 8/20 0.73
EGFR P00533 3/20 0.73
PRKACA P17612 1/20 0.73
PRKACG P22612 1/20 0.73
PRKACB P22694 1/20 0.73
PIK3CA P42336 1/20 0.69
PIK3CG P48736 1/20 0.69
PDGFRB P09619 5/20 0.69
PDGFRA P16234 5/20 0.69
PRKD3 O94806 2/20 0.63
PRKCG P05129 2/20 0.63
PRKCB P05771 2/20 0.63
PRKCH P24723 2/20 0.63
PRKCI P41743 2/20 0.63
PRKCE Q02156 2/20 0.63
PRKCQ Q04759 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469833 0.89 ABL1 (0.81) ABL1BCRPRKCASRCPRKCD
SCHEMBL4084867 0.87 ABL1 (0.77) ABL1BCRPRKCASRCPRKCD
SCHEMBL7467324 0.86 ABL1 (0.76) ABL1BCRPRKCASRCPRKCD
SCHEMBL29618427 0.84 ABL1 (0.85) ABL1BCRPRKCASRCPRKCD
SCHEMBL6254782 0.84 ABL1 (1.00) ABL1BCRPRKCASRCPRKCD
SCHEMBL7461678 0.84 ABL1 (0.73) ABL1BCRPRKCASRCPRKCD
SCHEMBL1465 0.84 ABL1 (1.00) ABL1BCRPRKCASRCPRKCD
SCHEMBL7474612 0.84 PIK3CG (0.76) ABL1BCRPRKCASRCPRKCD
SCHEMBL17070834 0.84 ABL1 (0.72) ABL1BCRPRKCASRCPRKCD
SCHEMBL7528647 0.84 ABL1 (0.72) ABL1BCRPRKCASRCPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098473-A1 REAGENTS AND METHODS FOR ANALYSIS OF PROTEINS AND METABOLITES TARGETED BY COVALENT PROBES DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-05-31 WO disclosed
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed