SCHEMBL7476833

SCHEMBL7476833

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCNC(=O)OC(C)(C)C)ccc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
HTT P42858 1/20 0.40
KDM4E B2RXH2 4/20 0.40
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
GPBAR1 Q8TDU6 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ATM Q13315 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966619 0.87 CA12 (0.41) ALDH1A1CA12CA1CA2CA9
SCHEMBL7373593 0.86 ALDH1A1 (0.43) ALDH1A1HTTKDM4ELMNAMAPT
SCHEMBL7427859 0.85 GPBAR1 (0.38) ALDH1A1CA12CA1CA2CA9
SCHEMBL7422214 0.85 MAPT (0.43) ALDH1A1HTTKDM4ECA12CA1
SCHEMBL7590287 0.85 MAPT (0.38) ALDH1A1HTTKDM4EL3MBTL1ATM
SCHEMBL7377107 0.84 ALDH1A1 (0.43) ALDH1A1HTTKDM4EATMMAPT
SCHEMBL7345680 0.84 ALDH1A1 (0.43) ALDH1A1HTTKDM4ELMNAMAPT
SCHEMBL7376935 0.82 ALDH1A1 (0.43) ALDH1A1HTTKDM4ELMNAMAPT
SCHEMBL7338369 0.81 TNF (0.42) ALDH1A1HTTKDM4EL3MBTL1LMNA
SCHEMBL7376973 0.80 ALDH1A1 (0.43) ALDH1A1HTTKDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed