SCHEMBL7476863

SCHEMBL7476863

Cc1ccc2c(c1)C(=O)N(CCCCN1CCN(c3ccccn3)CC1)C(CCl)=CO2

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.51
HTR1A P08908 4/20 0.51
DRD2 P14416 4/20 0.51
HTR2A P28223 3/20 0.51
HTR7 P34969 3/20 0.51
HTR6 P50406 2/20 0.51
GRIN1 Q05586 1/20 0.46
GRIN2B Q13224 1/20 0.46
DRD4 P21917 2/20 0.46
HTR2C P28335 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
DRD3 P35462 2/20 0.45
DRD1 P21728 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470711 0.93 KCNH2 (0.51) KCNH2HTR1ADRD2HTR2AHTR7
SCHEMBL7470291 0.90 HTR1A (0.49) KCNH2HTR1ADRD2HTR2AHTR7
SCHEMBL7463338 0.85 DRD4 (0.46) DRD2DRD4ADRA1DADRA1AADRA1B
SCHEMBL7469333 0.82 SIGMAR1 (0.47) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7469040 0.82 DRD4 (0.50) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7472411 0.82 HTR1A (0.58) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7467221 0.81 HTR1A (0.57) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7470410 0.81 HTR1A (0.53) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7467334 0.81 HTR1A (0.65) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL7472431 0.80 HTR7 (0.52) KCNH2HTR1ADRD2HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755930-B1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LTD (JP) 2002-07-31 EP disclosed
US-6337397-B1 A BENZOXAZEPINE DERIVATIVE FOR TREATMENT OF ANXIETY NEUROSIS, PHOBIAS, OBSESSIVE-COMPULSIVE DISORDERS, SCHIZOPHRENIA, POST-CARDIAC TRAUMA STRESS DISORDERS, DEPRESSION DISORDERS, PSYCHOSOMATIC DISORDERS AND OTHER PSYCHONEUROTIC DISORDERS, SUNTORY LIMITED (JP) 2002-01-08 US disclosed
US-6187769-B1 Benzoxazepine derivatives and their salts and medicaments containing the same SUNTORY LIMITED (JP) 2001-02-13 US disclosed
EP-0755930-A1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LIMITED (JP) 1997-01-29 EP disclosed