SCHEMBL7477292

SCHEMBL7477292

CCCCCNc1ncc(-c2ccc(OC(F)(F)F)cc2OC)nc1CC

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 9/20 0.52
ABL1 P00519 2/20 0.39
ADORA3 P0DMS8 3/20 0.38
BRD4 O60885 1/20 0.36
KCNH2 Q12809 1/20 0.35
RUNX1 Q01196 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201786 0.83 CRHR1 (0.60) CRHR1BRD4
SCHEMBL6203614 0.83 CRHR1 (0.70) CRHR1BRD4
SCHEMBL5415730 0.82 CRHR1 (0.72) CRHR1
SCHEMBL7477682 0.81 CRHR1 (0.57) CRHR1BRD4
SCHEMBL6201263 0.79 CRHR1 (0.62) CRHR1BRD4TLR8TLR7
SCHEMBL7482495 0.79 CRHR1 (0.41) CRHR1ABL1BRD4KCNH2RUNX1
SCHEMBL7477918 0.77 CRHR1 (0.70) CRHR1
SCHEMBL7480917 0.76 CRHR1 (0.51) CRHR1ABL1ADORA3RUNX1
SCHEMBL7476681 0.76 CRHR1 (0.58) CRHR1ADORA3BRD4
SCHEMBL7473622 0.76 CRHR1 (0.58) CRHR1BRD4TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP disclosed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO disclosed