SCHEMBL7477918

SCHEMBL7477918

CCCCCNc1nc(CC)c(-c2ccc(OC)cc2OC(F)(F)F)nc1CC

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 18/20 0.70
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
MERTK Q12866 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479339 0.88 CRHR1 (0.54) CRHR1
SCHEMBL6201786 0.86 CRHR1 (0.60) CRHR1
SCHEMBL7478694 0.85 CRHR1 (0.69) CRHR1
SCHEMBL6203614 0.85 CRHR1 (0.70) CRHR1
SCHEMBL7477682 0.84 CRHR1 (0.57) CRHR1ALDH1A1
SCHEMBL7480941 0.82 CRHR1 (0.68) CRHR1
SCHEMBL6075409 0.82 CRHR1 (1.00) CRHR1
SCHEMBL7606978 0.82 CRHR1 (0.59) CRHR1
SCHEMBL7474501 0.82 CRHR1 (0.59) CRHR1
SCHEMBL7477860 0.81 CRHR1 (0.53) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed