SCHEMBL7477383

SCHEMBL7477383

CCCCCNc1nc(CC)c(-c2ccc3ccccc3c2)nc1CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOAT1 P35610 2/20 0.38
EPHX1 P07099 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
TRIM58 Q8NG06 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
S1PR2 O95136 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KCNH3 Q9ULD8 1/20 0.37
MAOA P21397 3/20 0.37
MAOB P27338 2/20 0.37
RAB9A P51151 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169750 0.80 KDM4E (0.40) KDM4EALDH1A1
SCHEMBL6074922 0.77 CRHR1 (0.54)
SCHEMBL7469231 0.71 TLR8 (0.41) KCNH3TLR8
SCHEMBL7474934 0.71 CRHR1 (0.50)
SCHEMBL7478694 0.69 CRHR1 (0.69)
SCHEMBL7481401 0.69 CRHR1 (0.65) TLR7ALDH1A1
SCHEMBL6169536 0.69 CRHR1 (0.41) TLR7KDM4EALDH1A1
SCHEMBL9902645 0.69 SOAT1 (0.44) SOAT1EPHX1L3MBTL1KCNH3RAB9A
SCHEMBL8589161 0.69 EPHX1 (0.60) EPHX1TLR7LMNASMN1; SMN2KDM4E
SCHEMBL7477860 0.68 CRHR1 (0.53) KCNH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed