SCHEMBL7477593

SCHEMBL7477593

O=C1c2ccc(O)cc2C(=O)N1Nc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.46
ESR2 Q92731 6/20 0.46
CYP1A2 P05177 1/20 0.46
LMNA P02545 4/20 0.41
ANPEP P15144 2/20 0.41
DPP4 P27487 2/20 0.41
APP P05067 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
STAT3 P40763 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAOA P21397 1/20 0.39
UGT1A1 P22309 1/20 0.39
MAOB P27338 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7481106 0.98 ESR1 (0.45) ESR1ESR2CYP1A2LMNAANPEP
SCHEMBL7481797 0.86 STAT3 (0.52) ESR1ESR2CYP1A2LMNAAPP
SCHEMBL7486935 0.80 CASP6 (0.51) CYP1A2LMNATDP1MAOAMAOB
Hydrochloric Acid SCHEMBL7483427 0.80 CYP1A2 (0.45) CYP1A2LMNAALDH1A1MAPK1STAT3
SCHEMBL7485009 0.80 CYP1A2 (0.71) CYP1A2LMNAALDH1A1GAAMAPT
SCHEMBL7481564 0.78 STAT3 (0.45) ESR1ESR2LMNAANPEPDPP4
SCHEMBL7479666 0.78 APP (0.46) CYP1A2LMNAAPPALDH1A1MAPT
Hydrochloric Acid SCHEMBL7485356 0.77 APP (0.45) CYP1A2LMNAAPPALDH1A1MAPT
Hydrochloric Acid SCHEMBL7475918 0.76 STAT3 (0.43) ESR1ESR2LMNAANPEPDPP4
Hydrochloric Acid SCHEMBL7475915 0.76 STAT3 (0.43) ESR1ESR2LMNAANPEPDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed