SCHEMBL7481797

SCHEMBL7481797

O=C1c2ccc(Br)cc2C(=O)N1Nc1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP1A2 P05177 1/20 0.47
MAPT P10636 3/20 0.47
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
APP P05067 1/20 0.42
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.41
S100A4 P26447 1/20 0.40
LMNA P02545 3/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477593 0.86 ESR1 (0.46) STAT3NPSR1CYP1A2MAPTESR1
Hydrochloric Acid SCHEMBL7481106 0.84 ESR1 (0.45) STAT3NPSR1CYP1A2MAPTESR1
Hydrochloric Acid SCHEMBL7483427 0.81 CYP1A2 (0.45) STAT3NPSR1CYP1A2MAPTLMNA
SCHEMBL7485009 0.81 CYP1A2 (0.71) CYP1A2MAPTNPC1LMNACA1
SCHEMBL7479666 0.79 APP (0.46) CYP1A2MAPTAPPPOLBLMNA
Hydrochloric Acid SCHEMBL7485356 0.78 APP (0.45) CYP1A2MAPTAPPPOLBLMNA
SCHEMBL12443053 0.76 LMNA (0.71) STAT3NPSR1MAPTPOLBLMNA
SCHEMBL14322059 0.72 CYP1A2 (0.74) NPSR1CYP1A2MAPTAPPNPC1
SCHEMBL22743012 0.68 CYP1A2 (0.67) NPSR1CYP1A2MAPTCA1KMT2A
SCHEMBL1783796 0.67 APP (0.66) MAPTESR1ESR2APPPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed