SCHEMBL7478121

SCHEMBL7478121

COc1ccc2c(c1O)CN(Nc1ccncc1)CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 9/20 0.44
F3 P13726 5/20 0.44
DRD2 P14416 4/20 0.44
BCHE P06276 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CASP1 P29466 1/20 0.42
CYP2C19 P33261 1/20 0.42
APAF1 O14727 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.38
HCRTR2 O43614 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
ERN1 O75460 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7473644 0.99 DRD1 (0.43) DRD1F3DRD2BCHEKDM4E
SCHEMBL7482205 0.82 DRD2 (0.46) DRD1DRD2DRD3LIPE
SCHEMBL7477780 0.81 DRD1 (0.36) DRD1F3DRD2MEN1KMT2A
Hydrochloric Acid SCHEMBL7480606 0.81 DRD1 (0.36) DRD1F3DRD2MEN1KMT2A
SCHEMBL7489742 0.80 MEN1 (0.39) DRD2MEN1KMT2AHCRTR2ALDH1A1
SCHEMBL7484619 0.80 BCHE (0.38) DRD1F3DRD2BCHEMEN1
SCHEMBL7476993 0.78 DRD3 (0.52) DRD1DRD2KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL7474283 0.77 DRD3 (0.51) DRD1DRD2KDM4EMEN1KMT2A
SCHEMBL7476937 0.77 CYP19A1 (0.42) DRD1DRD2KDM4ELMNACYP1A2
SCHEMBL7487024 0.77 ALDH1A1 (0.38) MEN1KMT2AALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed