SCHEMBL7477780

SCHEMBL7477780

COc1ccc(O)c2c1CN(Nc1ccncc1)CC2

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.36
HTR1A P08908 2/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
ACHE P22303 1/20 0.35
KCNMA1 Q12791 1/20 0.33
DRD3 P35462 2/20 0.33
DRD4 P21917 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP19A1 P11511 1/20 0.32
F3 P13726 1/20 0.32
DRD2 P14416 1/20 0.32
DRD5 P21918 1/20 0.32
JAK2 O60674 1/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7480606 0.99 DRD1 (0.36) DRD1HTR1AMEN1KMT2AALDH1A1
SCHEMBL7487024 0.85 ALDH1A1 (0.38) MEN1KMT2AALDH1A1PKMKCNMA1
SCHEMBL7476937 0.85 CYP19A1 (0.42) DRD1MEN1KMT2AALDH1A1PKM
SCHEMBL7478121 0.81 DRD1 (0.44) DRD1MEN1KMT2AALDH1A1PKM
SCHEMBL7482604 0.81 KCNMA1 (0.33) MEN1KMT2AKCNMA1JAK2
Bromide SCHEMBL7473644 0.81 DRD1 (0.43) DRD1MEN1KMT2AALDH1A1PKM
Bromide SCHEMBL7475766 0.80 KCNMA1 (0.32) MEN1KMT2AKCNMA1JAK2
SCHEMBL7482205 0.79 DRD2 (0.46) DRD1DRD3CYP19A1DRD2DRD5
SCHEMBL7478156 0.78 CHRNA7 (0.42) HTR1AMEN1KMT2AALDH1A1TSHR
SCHEMBL7478986 0.78 CYP1A2 (0.30) HTR1AMEN1KMT2APKMKCNMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed