SCHEMBL7478252

SCHEMBL7478252

CC(C)(C)OC(=O)N1CCc2ccc(N3CCN(CCC(=O)NC(CC(=O)O)c4cccnc4)C3=O)cc2CC1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.47
ITGA2B P08514 7/20 0.47
ITGAV P06756 13/20 0.45
CYP3A4 P08684 1/20 0.39
CYP3A5 P20815 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468971 0.85 ITGB3 (0.42) ITGB3ITGA2BITGAV
SCHEMBL7474864 0.84 TMEM97 (0.39)
Trifluoroacetic Acid SCHEMBL7476025 0.83 ITGB3 (0.53) ITGB3ITGA2BITGAV
SCHEMBL7473247 0.80 NR1H2 (0.47)
SCHEMBL7481405 0.79 NR1H2 (0.42) ITGB3ITGA2B
SCHEMBL7468291 0.78 NR1H2 (0.38)
SCHEMBL7419930 0.75 NR1H2 (0.49)
Trifluoroacetic Acid SCHEMBL7480684 0.74 ITGB3 (0.49) ITGB3ITGA2BITGAV
SCHEMBL7468540 0.74 ITGB3 (0.39) ITGB3ITGA2BITGAV
SCHEMBL7469768 0.74 MAPT (0.41) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed