SCHEMBL7479718

SCHEMBL7479718

O=C(O)Oc1cccc2c1C(=O)c1ccccc1-2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
MAPT P10636 5/20 0.56
LMNA P02545 3/20 0.56
TTR P02766 3/20 0.50
NPC1 O15118 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KCNA3 P22001 1/20 0.46
TOP1 P11387 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
USP2 O75604 2/20 0.44
HTT P42858 2/20 0.44
ABCC4 O15439 1/20 0.44
TP53 P04637 1/20 0.44
HSP90AA1 P07900 1/20 0.44
CHRM2 P08172 1/20 0.44
HSP90AB1 P08238 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23212346 0.93 TTR (0.57) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL1727899 0.91 TTR (0.54) ALDH1A1MAPTLMNATTRL3MBTL1
SCHEMBL7109053 0.91 ALDH1A1 (0.51) ALDH1A1MAPTLMNATTRL3MBTL1
SCHEMBL27961252 0.87 TOP1 (0.46) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL5306728 0.87 MAPT (0.57) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL6036890 0.86 ALDH1A1 (0.51) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL5311970 0.81 EGFR (0.67) ALDH1A1MAPTLMNATTRL3MBTL1
SCHEMBL10883271 0.79 MAPT (0.52) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL8612875 0.79 MAPT (0.63) ALDH1A1MAPTLMNATTRNPC1
SCHEMBL11565971 0.79 MAPT (0.50) ALDH1A1MAPTLMNANPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1429768-B1 NOVEL MEDICAMENTS FOR INHALATION BOEHRINGER INGELHEIM PHARMA (DE) 2016-11-16 EP claimed
EP-0869947-B1 BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2002-10-23 EP claimed
EP-1429768-B1 NOVEL MEDICAMENTS FOR INHALATION BOEHRINGER INGELHEIM PHARMA (DE) 2016-11-16 EP disclosed