SCHEMBL7479940

SCHEMBL7479940

O=C1C=NCc2ccccc2N1CCCC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.40
HTR2A P28223 3/20 0.36
ADRA2B P18089 3/20 0.35
ADRA2C P18825 3/20 0.35
ADRA2A P08913 1/20 0.35
DRD2 P14416 7/20 0.34
DRD3 P35462 7/20 0.34
DRD5 P21918 3/20 0.34
HTR7 P34969 7/20 0.34
CHRM2 P08172 5/20 0.34
CHRM1 P11229 5/20 0.34
CHRM3 P20309 5/20 0.34
HTR1A P08908 5/20 0.34
CHRM4 P08173 4/20 0.34
CHRM5 P08912 4/20 0.34
DRD4 P21917 4/20 0.34
HRH1 P35367 3/20 0.34
SLC6A2 P23975 3/20 0.34
SLC22A2 O15244 2/20 0.34
SLC22A1 O15245 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246923 0.81 ADRA2B (0.40) SCN9AHTR2AADRA2BADRA2CADRA2A
SCHEMBL7248746 0.80 GSK3A (0.51) ADRA2BADRA2CADRA2ADRD2DRD3
SCHEMBL7241777 0.78 SMN1; SMN2 (0.49) HTR2ADRD2DRD3HTR1AHRH1
SCHEMBL7241537 0.77 ALDH1A1 (0.52) DRD3HTR7HTR1AHRH1SLC6A4
SCHEMBL7242765 0.77 GSK3A (0.49) ADRA2BADRA2CADRA2ADRD2DRD3
SCHEMBL7479946 0.76 SCN9A (0.40) SCN9AHTR2AADRA2BADRA2CADRA2A
SCHEMBL7247950 0.76 ADRA2A (0.44) ADRA2BADRA2CADRA2ADRD2DRD3
SCHEMBL7241382 0.76 ADRA2A (0.40) SCN9AADRA2BADRA2CADRA2ADRD2
SCHEMBL7248585 0.75 ACHE (0.40) SCN9ADRD2DRD3HTR7CHRM2
SCHEMBL11883909 0.75 CYP1A2 (0.41) ADRA2BADRA2CADRA2AADRA1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951466-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP claimed
WO-1998028268-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 1998-07-02 WO claimed