SCHEMBL7480268

SCHEMBL7480268

CC(C)(C)OC(=O)Nc1cccc(-c2nsc3nc4ccccc4n23)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.46
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
ACSS2 Q9NR19 1/20 0.38
MAP3K5 Q99683 3/20 0.37
TGFBR1 P36897 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LCK P06239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479244 0.82 BRD4 (0.52) BRD4OPRM1OPRD1OGFRL1ACSS2
SCHEMBL29394473 0.71 LCK (0.47) NPC1RAB9ASMN1; SMN2MEN1GAA
SCHEMBL7480580 0.71 CSNK1A1 (0.39) NPC1RAB9ATP53SMN1; SMN2GAA
SCHEMBL533505 0.69 RAB9A (0.62) NPC1RAB9ATP53SMN1; SMN2MEN1
SCHEMBL31151002 0.69 RAB9A (0.62) NPC1RAB9ATP53SMN1; SMN2MEN1
SCHEMBL7473909 0.69 CTSD (0.47) NPC1RAB9ATP53SMN1; SMN2MEN1
SCHEMBL23582507 0.68 SCN9A (0.52) SCN9A
SCHEMBL7486557 0.67 SMN1; SMN2 (0.43) BRD4NPC1RAB9ATP53SMN1; SMN2
SCHEMBL1721390 0.67 SCN9A (0.54) SMN1; SMN2ALDH1A1SCN9A
SCHEMBL7474969 0.67 DRD2 (0.54) NPC1RAB9ATP53SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-B1 PROTON PUMP INHIBITOR APOTEX INC (CA) 2002-05-15 EP disclosed
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed
US-6093738-A IMIDAZO(1,2-D)-THIADIAZOLE COMPOUNDS; PEPTIC ULCER TREATMENT KARIMIAN KHASHAYAR (CA) 2000-07-25 US disclosed