SCHEMBL7482091

SCHEMBL7482091

CCCCCOc1nc(CC)c(-c2ccc(C(F)(F)F)cc2C(F)(F)F)nc1CC

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 8/20 0.43
PDE2A O00408 2/20 0.35
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TRPV3 Q8NET8 2/20 0.33
SLC9A5 Q14940 1/20 0.32
PPARD Q03181 1/20 0.32
PTGES O14684 1/20 0.32
ALOX5 P09917 1/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480028 0.87 CRHR1 (0.47) CRHR1
SCHEMBL5411905 0.81 CRHR1 (0.58) CRHR1ABCC8KCNJ11TRPV3SLC9A5
SCHEMBL5414396 0.80 CRHR1 (0.45) CRHR1ABCC8KCNJ11TRPV3SLC9A5
SCHEMBL7473334 0.79 CRHR1 (0.45) CRHR1
SCHEMBL5412069 0.79 CRHR1 (0.51) CRHR1ABCC8KCNJ11TRPV3
SCHEMBL6201986 0.77 CRHR1 (0.39) CRHR1
SCHEMBL6200122 0.76 CRHR1 (0.47) CRHR1
SCHEMBL7483586 0.74 TLR8 (0.41) CRHR1PDE2A
SCHEMBL7479299 0.74 CRHR1 (0.65) CRHR1
SCHEMBL7474501 0.73 CRHR1 (0.59) CRHR1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed