SCHEMBL7483348

SCHEMBL7483348

c1ccc2nc(COc3ccc4c(c3)CCCN4)ccc2c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.60
CYSLTR1 Q9Y271 7/20 0.53
CYSLTR2 Q9NS75 3/20 0.53
GPBAR1 Q8TDU6 6/20 0.52
ALOX5AP P20292 3/20 0.52
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7532657 0.99 PDE10A (0.58) PDE10ACYSLTR1CYSLTR2GPBAR1ALOX5AP
SCHEMBL8140420 0.83 PDE10A (0.49) PDE10ACYSLTR1CYSLTR2
SCHEMBL8801873 0.82 MAOB (0.58) PDE10ACYSLTR1CYSLTR2ALOX5AP
SCHEMBL8129843 0.82 CYSLTR1 (0.53) PDE10ACYSLTR1CYSLTR2GPBAR1
SCHEMBL8801610 0.81 MAOA (0.56) CYSLTR1CYSLTR2GPBAR1
SCHEMBL6421129 0.78 MAOA (0.64)
SCHEMBL8801952 0.78 MAOA (0.62) PDE10ACYSLTR1CYSLTR2GPBAR1ALOX5AP
SCHEMBL10512475 0.77 PDE10A (0.77) PDE10ACYSLTR1CYSLTR2GPBAR1CYP1A2
SCHEMBL14302687 0.77 PDE10A (0.44) PDE10ACYSLTR1GPBAR1ALOX5APCYP1A2
SCHEMBL8801596 0.76 PDE10A (0.53) PDE10ACYSLTR1CYSLTR2GPBAR1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210343-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS AstraZeneca AB (SE) 2002-06-05 EP disclosed
WO-2001012187-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS ASTRAZENECA AB (SE) 2001-02-22 WO disclosed