SCHEMBL7484205

SCHEMBL7484205

CNN1CC[C@H](c2cncc(C(F)(F)F)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 1/20 0.36
HDAC4 P56524 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
DRD2 P14416 1/20 0.35
IDH1 O75874 1/20 0.35
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNB3 Q05901 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103958 1.00 PROKR1 (0.36) PROKR1HDAC4CYP11B1CYP11B2DRD2
SCHEMBL7101655 0.82 RIPK1 (0.38) HDAC4
SCHEMBL7103719 0.82 RIPK1 (0.38) HDAC4
SCHEMBL7097543 0.77 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3
SCHEMBL7487273 0.77 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3
SCHEMBL7101838 0.76 CHRNB4 (0.39) DRD2CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7101149 0.76 CHRNA3 (0.54) DRD2CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7102542 0.76 CHRNB4 (0.39) DRD2CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7099212 0.76 CHRNA3 (0.54) DRD2CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7098415 0.74 JAK2 (0.37) HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed