SCHEMBL748640

SCHEMBL748640

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)Oc2cc(F)cc3c2NCCC3)cc1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.32
CDK8 P49336 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
TACR2 P21452 1/20 0.32
TACR1 P25103 1/20 0.32
LMNA P02545 2/20 0.31
MAPK1 P28482 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
MAPT P10636 2/20 0.31
TP53 P04637 2/20 0.31
DHODH Q02127 2/20 0.31
NR1H4 Q96RI1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SIGMAR1 Q99720 4/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL749783 0.99 TACR3 (0.32) TACR3CDK8CLK4TACR2TACR1
SCHEMBL751895 0.92 DHODH (0.33) CDK8CLK4TACR2TACR1LMNA
SCHEMBL747960 0.91 CDK8 (0.32) CDK8CLK4TACR2TACR1LMNA
Hydrochloric Acid SCHEMBL750002 0.91 DHODH (0.33) CDK8CLK4TACR2TACR1LMNA
SCHEMBL748805 0.91 MAPT (0.36) LMNATRPV1MAPTTP53DHODH
Hydrochloric Acid SCHEMBL748195 0.91 CDK8 (0.32) CDK8CLK4TACR2TACR1LMNA
SCHEMBL750950 0.89 SRC (0.36) CDK8CLK4LMNATRPV1MAPT
SCHEMBL746629 0.88 WDR5 (0.33) LMNATRPV1MAPTTP53DHODH
Hydrochloric Acid SCHEMBL751875 0.88 SRC (0.36) CDK8CLK4LMNATRPV1MAPT
SCHEMBL749615 0.87 MAPT (0.35) LMNATRPV1MAPTTP53DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed