SCHEMBL747960

SCHEMBL747960

Cc1cc2c(c(OC(=O)N(CCc3ccc(Cl)c(Cl)c3)Cc3ccc(C(C)(C)C)cc3)c1)NCCC2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
DHODH Q02127 2/20 0.31
NR1H4 Q96RI1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SIGMAR1 Q99720 7/20 0.31
TP53 P04637 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2D6 P10635 2/20 0.31
TSHR P16473 2/20 0.31
ESRRB O95718 1/20 0.31
ESRRG P62508 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL748195 0.99 CDK8 (0.32) CDK8CLK4TRPV1DHODHNR1H4
SCHEMBL751895 0.93 DHODH (0.33) CDK8CLK4TRPV1DHODHNR1H4
Hydrochloric Acid SCHEMBL750002 0.92 DHODH (0.33) CDK8CLK4TRPV1DHODHNR1H4
SCHEMBL748640 0.91 TACR3 (0.32) CDK8CLK4TRPV1DHODHNR1H4
Hydrochloric Acid SCHEMBL749783 0.91 TACR3 (0.32) CDK8CLK4TRPV1DHODHNR1H4
SCHEMBL750950 0.89 SRC (0.36) CDK8CLK4TRPV1DHODHNR1H4
Hydrochloric Acid SCHEMBL751875 0.89 SRC (0.36) CDK8CLK4TRPV1DHODHNR1H4
SCHEMBL750907 0.89 MAPT (0.35) TRPV1DHODHALDH1A1LMNAMAPT
SCHEMBL746654 0.86 OPRM1 (0.34) TRPV1NR1H4ALDH1A1MAPTSIGMAR1
SCHEMBL746629 0.86 WDR5 (0.33) TRPV1DHODHALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed