SCHEMBL7487333

SCHEMBL7487333

COc1ccc(S(=O)(=O)N(Cc2cccnc2)C[C@@H](C)S)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 11/20 0.57
MMP2 P08253 3/20 0.57
ALDH1A1 P00352 2/20 0.57
CXCR3 P49682 2/20 0.55
PDE4A P27815 2/20 0.54
PDE4B Q07343 2/20 0.54
PDE4C Q08493 2/20 0.54
PDE4D Q08499 2/20 0.54
RAB9A P51151 1/20 0.52
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
ALOX12 P18054 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MMP13 P45452 7/20 0.49
MMP1 P03956 6/20 0.49
ADAM17 P78536 5/20 0.49
PTGES O14684 1/20 0.47
TAS2R14 Q9NYV8 1/20 0.47
TAS2R8 Q9NYW2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6321605 1.00 MMP9 (0.57) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL6323674 0.89 MMP9 (0.60) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL6323932 0.86 TAS2R14 (0.62) ALDH1A1CXCR3LMNAPTGESTAS2R14
SCHEMBL6326217 0.83 MMP9 (0.57) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL26770427 0.81 ALDH1A1 (0.73) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL6321598 0.80 MMP9 (0.63) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL6321600 0.80 MMP9 (0.63) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL26770391 0.80 MMP9 (0.55) MMP9MMP2ALDH1A1CXCR3PDE4A
SCHEMBL1169467 0.78 TAS2R14 (0.79) ALDH1A1CXCR3PTGESTAS2R14TAS2R8
SCHEMBL7340409 0.78 ALDH1A1 (0.75) MMP9MMP2ALDH1A1CXCR3MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939629-A4 THIOL SULFONAMIDE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2002-07-17 EP disclosed
EP-0939629-A1 THIOL SULFONAMIDE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003166-A1 THIOL SULFONAMIDE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed