SCHEMBL7488479

SCHEMBL7488479

CC(C)C[C@H](NC(=O)c1ccccc1-c1csc(N2CCNCC2)n1)C(=O)NC1(C#N)CC1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSL P07711 14/20 0.52
CTSK P43235 10/20 0.50
CTSS P25774 8/20 0.50
CTSB P07858 6/20 0.50
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606091 0.86 CTSK (0.60) CTSLCTSKCTSSCTSB
SCHEMBL6183387 0.86 CTSK (0.60) CTSLCTSKCTSSCTSB
SCHEMBL7451288 0.84 CTSL (0.51) CTSLCTSKCTSSCTSB
SCHEMBL7427146 0.84 CTSL (0.49) CTSLCTSKCTSSCTSB
SCHEMBL6184402 0.78 CTSK (0.61) CTSLCTSKCTSSCTSBKCNH2
SCHEMBL4759913 0.77 CTSK (0.78) CTSLCTSKCTSSCTSBKCNH2
SCHEMBL4760512 0.77 CTSK (0.78) CTSLCTSKCTSSCTSBKCNH2
SCHEMBL7650778 0.75 CTSL (0.59) CTSLCTSKCTSSCTSB
SCHEMBL7488490 0.74 CTSK (0.48) CTSLCTSKCTSSCTSBKCNH2
SCHEMBL6183633 0.74 CTSL (0.59) CTSLCTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed