SCHEMBL7489125

SCHEMBL7489125

C=C(C(=O)OC)N(c1ccccc1Cc1ccccc1NC(=O)c1cccnc1)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.49
ALDH1A1 P00352 4/20 0.48
MAPT P10636 3/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 2/20 0.48
HPGD P15428 2/20 0.47
HTT P42858 1/20 0.47
POLB P06746 2/20 0.46
AVPR1B P47901 1/20 0.45
MEN1 O00255 1/20 0.45
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPC1 O15118 1/20 0.43
PKM P14618 2/20 0.42
LMNA P02545 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610253 0.85 ABCB1 (0.51) ABCB1ALDH1A1MAPTKMT2AGAA
SCHEMBL7489133 0.81 ABCB1 (0.47) ABCB1ALDH1A1MAPTKMT2AGAA
SCHEMBL6610090 0.75 SNCA (0.47) MAPTKMT2APOLBAVPR1BMEN1
SCHEMBL5656436 0.75 LMNA (0.48) MAPTKMT2APOLBNPC1LMNA
SCHEMBL8628089 0.72 MAPT (0.60) ALDH1A1MAPTKMT2AGAAPOLB
SCHEMBL6611082 0.71 LMNA (0.42) MAPTKMT2APOLBLMNAKEAP1
SCHEMBL6609938 0.70 MAPT (0.48) ALDH1A1MAPTKMT2AHTTPOLB
SCHEMBL6612494 0.70 TAS2R14 (0.46) ABCB1ALDH1A1MAPTKMT2AHPGD
SCHEMBL6608937 0.70 MEN1 (0.47) ABCB1ALDH1A1MAPTKMT2AGAA
SCHEMBL6613518 0.69 ALDH1A1 (0.47) ALDH1A1MAPTHPGDSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147095-A1 2, 3, 4, 5-TETRAHYDRO-1H-[1, 4] BENZODIAZEPINE-3-HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS American Cyanamid Company (US) 2001-10-24 EP disclosed
WO-2000044730-A1 2,3,4,5-TETRAHYDRO-1H-[1,4]BENZODIAZEPINE-3-HYDROXAMIC ACID AS MATRIX METALLOPROTEINASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed