SCHEMBL749564

SCHEMBL749564

CC(C)(C)c1ccc(CN(CCc2ccc(F)cc2)C(=O)c2cc(Cl)cc3cccnc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
F7 P08709 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
SLC2A1 P11166 1/20 0.39
C5AR1 P21730 1/20 0.37
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ESRRG P62508 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL750788 0.88 OPRM1 (0.47) TP53MAPTF2F10F7
SCHEMBL12520898 0.79 TP53 (0.53) TP53MAPTSLC2A1C5AR1ESRRG
SCHEMBL3570656 0.78 TP53 (0.42) TP53MAPTF2F10F7
SCHEMBL3573203 0.77 RAF1 (0.40) TP53MAPTOPRM1OPRD1C5AR1
SCHEMBL747155 0.76 TP53 (0.38) TP53MAPTF2F10F7
SCHEMBL3581435 0.75 TP53 (0.41) TP53MAPTF2F10F7
Hydrochloric Acid SCHEMBL748268 0.75 TP53 (0.38) TP53MAPTF2F10F7
SCHEMBL12521008 0.74 TP53 (0.48) TP53MAPTSLC2A1ESRRGBCL2
SCHEMBL12521175 0.74 LPAR1 (0.41) TP53MAPTOPRM1OPRD1C5AR1
SCHEMBL12520957 0.74 TP53 (0.43) TP53MAPTF2F10F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed