SCHEMBL7498253

SCHEMBL7498253

Cc1ccc(C)c(-n2ccc(C)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.46
ALDH1A1 P00352 5/20 0.43
APOBEC3G Q9HC16 2/20 0.38
KDM4E B2RXH2 1/20 0.38
APOBEC3A P31941 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
MPI P34949 4/20 0.36
PHOSPHO1 Q8TCT1 4/20 0.36
PMM2 O15305 3/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
SLC18A3 Q16572 1/20 0.34
HCAR1 Q9BXC0 1/20 0.34
G6PD P11413 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270640 0.78 HSD17B10 (0.48) HSD17B10ALDH1A1KDM4ETDP1MPI
SCHEMBL645578 0.78 TP53 (0.39) HSD17B10ALDH1A1TDP1MPIPHOSPHO1
SCHEMBL7772481 0.77 TUBB4A (0.42) HSD17B10ALDH1A1KDM4ETDP1TSHR
SCHEMBL2750548 0.72 HSD17B10 (0.43) HSD17B10ALDH1A1KDM4ETDP1MPI
SCHEMBL23292676 0.71 MAPT (0.52) ALDH1A1KDM4ETSHRMEN1KMT2A
SCHEMBL11569176 0.71 IDO1 (0.44) HSD17B10ALDH1A1TDP1TSHRMEN1
SCHEMBL16141626 0.69 HSD17B10 (0.41) HSD17B10ALDH1A1APOBEC3GAPOBEC3ATDP1
SCHEMBL18850042 0.69 MGLL (0.43) HSD17B10ALDH1A1APOBEC3GKDM4ETDP1
Iodide SCHEMBL17509707 0.68 HSD17B10 (0.40) HSD17B10ALDH1A1APOBEC3GAPOBEC3ATDP1
SCHEMBL3310092 0.68 ALDH1A1 (0.52) HSD17B10ALDH1A1APOBEC3GKDM4EMPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265870-A1 NEW CCR5 MODULATORS: BENZIMIDAZOLES OR BENZOTRIAZOLES AstraZeneca AB (SE) 2002-12-18 EP disclosed
WO-2001066525-A1 NEW CCR5 MODULATORS: BENZIMIDAZOLES OR BENZOTRIAZOLES ASTRAZENECA AB (SE) 2001-09-13 WO disclosed