SCHEMBL7498541

SCHEMBL7498541

CC(C)(C)OC(=O)NCC12CN(c3cc4c(cc3F)c(=O)c(OC(=O)O)cn4C(C)(C)CF)CC1CCO2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.36
KDM4E B2RXH2 9/20 0.36
HPGD P15428 6/20 0.36
HSD17B10 Q99714 5/20 0.36
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
LMNA P02545 3/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
TOP2B Q02880 2/20 0.32
DRD3 P35462 1/20 0.32
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
TOP2A P11388 1/20 0.31
CYP2C9 P11712 1/20 0.31
BRD4 O60885 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
CYP2J2 P51589 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502083 0.96 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7494808 0.93 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7494670 0.93 KDM4E (0.35) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7843329 0.92 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL9211202 0.90 KDM4E (0.43) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9208089 0.89 LMNA (0.35) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7498548 0.89 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7847782 0.87 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDHSD17B10MEN1
Trifluoroacetic Acid SCHEMBL7501716 0.85 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7834705 0.85 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944385-B1 USE OF 7-(1-AMINOMETHYL-2-OXA-7-AZA-BICYCLO 3.3.0]OCT-7-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDONE CARBOXYLIC ACID DERIVATIVES FOR TREATING HELICOBACTER PYLORI INFECTIONS AND THE GASTRODUODENAL DISEASES ASSOCIATED THEREWITH BAYER AG (DE) 2002-10-16 EP disclosed