SCHEMBL7499057

SCHEMBL7499057

CCOC(=O)c1nc(-c2ccccc2)c(-c2ccc(S(N)(=O)=O)cc2)o1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
CA9 Q16790 6/20 0.54
CA12 O43570 5/20 0.54
PTGS2 P35354 6/20 0.50
PTGS1 P23219 4/20 0.50
NR4A2 P43354 3/20 0.50
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 1/20 0.47
RXRA P19793 2/20 0.47
RXRB P28702 2/20 0.47
RXRG P48443 1/20 0.47
ADORA3 P0DMS8 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
MT-CO2 P00403 1/20 0.46
LMNA P02545 1/20 0.46
CA3 P07451 1/20 0.46
ADRB2 P07550 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7505599 1.00 CA1 (0.58) CA1CA2CA9CA12PTGS2
SCHEMBL7500361 0.90 PTGS2 (0.62) CA1CA2CA9CA12PTGS2
SCHEMBL7501340 0.90 PTGS2 (0.62) CA1CA2CA9CA12PTGS2
SCHEMBL2117681 0.88 NR4A2 (0.63) NR4A2KMT2AALDH1A1HSD17B10RXRA
SCHEMBL7510938 0.87 NR4A2 (0.53) CA1CA2CA9CA12PTGS2
SCHEMBL7504069 0.87 NR4A2 (0.53) CA1CA2CA9CA12PTGS2
SCHEMBL8546268 0.83 NR4A2 (0.57) CA1CA2CA9CA12PTGS2
SCHEMBL8556797 0.83 ALDH1A1 (0.46) CA1CA2CA9CA12NR4A2
SCHEMBL8558012 0.83 CA1 (0.44) CA1CA2CA9CA12NR4A2
SCHEMBL7502759 0.83 NR4A2 (0.73) CA1CA2CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0699192-B1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-07-24 EP claimed
EP-0699192-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-06 EP claimed
WO-1994027980-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1994-12-08 WO claimed
EP-0699192-B1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-07-24 EP disclosed
EP-0699192-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-06 EP disclosed
WO-1994027980-A1 SUBSTITUTED OXAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1994-12-08 WO disclosed