SCHEMBL7499403

SCHEMBL7499403

CN1CC=C(c2ccc3cc(C(=O)N(C)C)[nH]c3c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
QDPR P09417 3/20 0.48
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
HRH4 Q9H3N8 4/20 0.40
ROCK2 O75116 2/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28421403 0.76 QDPR (0.49) QDPRHTR1DHTR1B
SCHEMBL7501974 0.73 QDPR (0.48) QDPRHTR1DHTR1B
SCHEMBL6739833 0.72 QDPR (0.56) QDPRHTR1DHTR1B
SCHEMBL9051846 0.71 AR (0.49) ROCK2
SCHEMBL6741293 0.71 QDPR (0.49) QDPRHTR1DHTR1B
SCHEMBL28422171 0.69 QDPR (0.55) QDPRHTR1DHTR1B
SCHEMBL31342570 0.68 ROCK2 (0.35) HRH4ROCK2CDK2
SCHEMBL22152424 0.68 HRH4 (0.55) HRH4
SCHEMBL7744453 0.66 QDPR (1.00) QDPRHTR1DHTR1B
SCHEMBL14845694 0.66 PIN1 (0.68) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196380-A2 INDOLES AND INDAZOLES FOR THE TREATMENT OF MIGRAINE NPS Allelix Corp. (CA) 2002-04-17 EP disclosed
WO-2001005758-A2 INDOLES AND INDAZOLES FOR THE TREATMENT OF MIGRAINE NPS ALLELIX CORP. (CA) 2001-01-25 WO disclosed