SCHEMBL7499837

SCHEMBL7499837

CCC(=O)N(c1ccccc1)[C@H](C(=O)OC(C)(C)C)C1CCCNC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
SLC6A2 P23975 6/20 0.36
SLC6A4 P31645 6/20 0.36
OPRM1 P35372 1/20 0.35
CPN1 P15169 1/20 0.34
CPB2 Q96IY4 1/20 0.34
SLC6A3 Q01959 5/20 0.34
CYP2D6 P10635 2/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHRM3 P20309 1/20 0.34
KCNH2 Q12809 1/20 0.34
TSHR P16473 1/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493966 1.00 KMT2A (0.36) KMT2AMAPTPKMSLC6A2SLC6A4
SCHEMBL7493957 1.00 KMT2A (0.36) KMT2AMAPTPKMSLC6A2SLC6A4
SCHEMBL7497433 0.90 KMT2A (0.35) KMT2AMAPTPKMSLC6A2SLC6A4
SCHEMBL7496627 0.89 AAK1 (0.37) MAPTPKMSLC6A2SLC6A4OPRM1
SCHEMBL7500612 0.89 HTT (0.34) KMT2ASLC6A2SLC6A4CPN1CPB2
SCHEMBL7505927 0.89 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3CYP2D6CHRNB2
SCHEMBL7966504 0.87 KMT2A (0.34) KMT2AMAPTPKMSLC6A2SLC6A4
SCHEMBL7500113 0.82 KMT2A (0.42) KMT2AMAPTPKMSLC6A2SLC6A4
SCHEMBL7496325 0.82 CACNA2D1 (0.41) KMT2ASLC6A2SLC6A4OPRM1SLC6A3
SCHEMBL7491286 0.82 ALDH1A1 (0.40) OPRM1CHRM3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002069895-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND METHODS OF USE THEREOF SEPRACOR, INC. (US) 2002-09-12 WO disclosed
EP-1187810-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND THEIR USE SEPRACOR, INC. (US) 2002-03-20 EP disclosed
WO-2001092226-A1 HETEROCYCLIC ANALGESIC COMPOUNDS AND METHOD OF USE THEREOF SEPRACOR, INC. (US) 2001-12-06 WO disclosed
WO-2000071518-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND THEIR USE SEPRACOR, INC. (US) 2000-11-30 WO disclosed