SCHEMBL7500612

SCHEMBL7500612

CC(C)(C)OC(=O)C(C1CCCNC1)N(C(=O)C1CC1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
CCR8 P51685 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
EPHX2 P34913 1/20 0.33
CPN1 P15169 1/20 0.33
CPB2 Q96IY4 1/20 0.33
SSTR1 P30872 1/20 0.32
SSTR4 P31391 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493966 0.89 KMT2A (0.36) KMT2ASLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7499837 0.89 KMT2A (0.36) KMT2ASLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7493957 0.89 KMT2A (0.36) KMT2ASLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7498061 0.88 SLC6A2 (0.38) KMT2ASLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7497433 0.85 KMT2A (0.35) KMT2ACCR8SLC6A2SLC6A4SLC6A3
SCHEMBL7966504 0.84 KMT2A (0.34) KMT2ACCR8SLC6A2SLC6A4SLC6A3
SCHEMBL7491286 0.82 ALDH1A1 (0.40) ALDH1A1NR1H4
SCHEMBL7496325 0.82 CACNA2D1 (0.41) KMT2AALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL7528853 0.81 POLB (0.43) KMT2ACCR8ALDH1A1LMNASLC6A2
SCHEMBL7505927 0.78 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3KCNH2CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002069895-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND METHODS OF USE THEREOF SEPRACOR, INC. (US) 2002-09-12 WO disclosed
EP-1187810-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND THEIR USE SEPRACOR, INC. (US) 2002-03-20 EP disclosed
WO-2000071518-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND THEIR USE SEPRACOR, INC. (US) 2000-11-30 WO disclosed