SCHEMBL7500221

SCHEMBL7500221

COC(=O)COc1ccc(C(=O)CN(C)C(=O)CCc2ccncc2)cc1OCC(=O)OC.O=C(O)CCc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.46
ITGA2B P08514 2/20 0.46
CNR2 P34972 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
FFAR1 O14842 2/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NOX1 Q9Y5S8 1/20 0.35
NAMPT P43490 1/20 0.35
ROCK2 O75116 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
ROCK1 Q13464 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009746 0.96 ITGB3 (0.45) ITGB3ITGA2BCNR2MEN1KMT2A
SCHEMBL7499998 0.90 ITGB3 (0.55) ITGB3ITGA2BCNR2MEN1KMT2A
SCHEMBL7368949 0.72 ITGB3 (0.50) ITGB3ITGA2BMEN1KMT2AALDH1A1
SCHEMBL7363023 0.71 ITGB3 (0.49) ITGB3ITGA2BMEN1KMT2AL3MBTL1
SCHEMBL8180044 0.70 ITGB3 (0.51) ITGB3ITGA2BMEN1KMT2AL3MBTL1
SCHEMBL7358969 0.68 KMT2A (0.67) MEN1KMT2AL3MBTL1CYP3A4CYP2C9
SCHEMBL7407172 0.67 KMT2A (0.50) ITGB3ITGA2BMEN1KMT2AL3MBTL1
SCHEMBL8012315 0.67 ITGB3 (0.52) ITGB3ITGA2BMEN1KMT2AL3MBTL1
SCHEMBL8641278 0.66 NPSR1 (0.36) MEN1KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL8633992 0.65 ALDH1A1 (0.55) MEN1KMT2ACYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677043-A4 1995-11-22 EP disclosed
EP-0677043-A1 PLATELET AGGREGATION INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-10-18 EP disclosed
WO-1994014775-A1 PLATELET AGGREGATION INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed