SCHEMBL7500962

SCHEMBL7500962

CC1(NCc2ccccc2)CCCNC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
CYP2D6 P10635 4/20 0.43
TSHR P16473 1/20 0.43
USP2 O75604 2/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37
HTR2A P28223 2/20 0.36
SSTR3 P32745 1/20 0.36
CYP1A2 P05177 1/20 0.36
CXCR4 P61073 1/20 0.36
SLC6A4 P31645 3/20 0.36
TACR1 P25103 2/20 0.36
CDK7 P50613 1/20 0.35
CCNH P51946 1/20 0.35
MNAT1 P51948 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608911 0.90 HTR2A (0.41) CYP3A4CYP2D6TSHRALDH1A1CYP2C9
SCHEMBL27800697 0.81 CYP3A4 (0.43) CYP3A4TSHRSSTR3KDM4EMAPT
SCHEMBL11039283 0.81 CYP3A4 (0.43) CYP3A4SSTR3KDM4EMAPT
SCHEMBL4604214 0.80 TACR1 (0.44) CYP3A4CYP2D6TSHRALDH1A1CYP2C9
SCHEMBL27893441 0.80 KDM4E (0.42) CYP3A4TSHRSSTR3SLC6A4KDM4E
Bromide SCHEMBL11037477 0.80 CYP3A4 (0.42) CYP3A4SSTR3KDM4EMAPT
SCHEMBL27890446 0.77 CYP3A4 (0.46) CYP3A4KDM4EMAPT
SCHEMBL4082174 0.76 CYP3A4 (0.41) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL15928065 0.73 IDO1 (0.39) CYP3A4CYP2D6TSHRHTR2ACXCR4
SCHEMBL14650073 0.73 CTSS (0.48) CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723545-B1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LAB (US) 2002-05-08 EP disclosed
EP-0871628-A1 QUINOLIZINONE TYPE COMPOUNDS Abbott Laboratories (US) 1998-10-21 EP disclosed
US-5726182-A TREATMENT OF BACTERIAL INFECTIONS ABBOTT LABORATORIES (US) 1998-03-10 US disclosed
US-5599816-A BACTERICIDE ABBOTT LABORATORIES (US) 1997-02-04 US disclosed
WO-1996039407-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-12-12 WO disclosed
US-5580872-A ADMINISTERING IN THE TREATMENT OF BACTERIAL INFECTIONS ABBOTT LABORATORIES (US) 1996-12-03 US disclosed
EP-0723545-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1996-07-31 EP disclosed
WO-1995010519-A1 QUINOLIZINONE TYPE COMPOUNDS ABBOTT LABORATORIES (US) 1995-04-20 WO disclosed