SCHEMBL7501140

SCHEMBL7501140

N[C@H]1C=CC=CN(CC(=O)O)C1=O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
APEX1 P27695 1/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31
RAB9A P51151 1/20 0.30
ACE P12821 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5066904 1.00 SMN1; SMN2 (0.38) SMN1; SMN2L3MBTL1APEX1CA12CA9
SCHEMBL11007720 0.68 SMN1; SMN2 (0.33) SMN1; SMN2L3MBTL1
SCHEMBL27451981 0.68 ALDH1A1 (0.34) SMN1; SMN2L3MBTL1APEX1CA12CA9
SCHEMBL7062477 0.68 SMN1; SMN2 (0.35) SMN1; SMN2L3MBTL1APEX1ACEDPP4
SCHEMBL7058422 0.68 SMN1; SMN2 (0.35) SMN1; SMN2L3MBTL1APEX1ACEDPP4
SCHEMBL27287079 0.67 TSHR (0.36) SMN1; SMN2L3MBTL1APEX1CA12CA9
SCHEMBL6347888 0.62 SMN1; SMN2 (0.33) SMN1; SMN2L3MBTL1ACE
SCHEMBL11513013 0.62
SCHEMBL28187140 0.60 SMN1; SMN2 (0.30) SMN1; SMN2L3MBTL1
SCHEMBL1133635 0.59 P2RX4 (0.41) SMN1; SMN2APEX1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932733-A INHIBITOR OF THROMBIN CORVAS INTERNATIONAL, INC. (US) 1999-08-03 US disclosed
EP-0765339-B1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES CONTAINING AN ARGININE MIMIC AS ENZYME INHIBITORS CORVAS INT INC (US) 1999-01-27 EP disclosed
EP-0765339-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES CONTAINING AN ARGININE MIMIC AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1997-04-02 EP disclosed
WO-1995035313-A1 3-AMINO-2-OXO-1-PIPERIDINEACETIC DERIVATIVES CONTAINING AN ARGININE MIMIC AS ENZYME INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1995-12-28 WO disclosed