SCHEMBL7508166

SCHEMBL7508166

COC(=O)CCCC(=O)c1ccc(OC)c(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.58
CYP1A2 P05177 4/20 0.51
CYP2C19 P33261 4/20 0.51
CYP2D6 P10635 1/20 0.51
HPGD P15428 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
RECQL P46063 1/20 0.48
KCNH2 Q12809 1/20 0.48
CTNNB1 P35222 2/20 0.48
WNT3A P56704 2/20 0.48
MAPT P10636 4/20 0.47
CYP3A4 P08684 2/20 0.47
KDM4E B2RXH2 1/20 0.47
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
ALOX12 P18054 2/20 0.46
KMT2A Q03164 2/20 0.46
RAB9A P51151 2/20 0.46
HTT P42858 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499557 0.83 L3MBTL1 (0.50) CYP1A2L3MBTL1MAPTTHRATHRB
SCHEMBL7506850 0.83 NPC1 (0.44) CYP1A2L3MBTL1MAPTTHRATHRB
SCHEMBL5729109 0.82 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL8416607 0.82 CTNNB1 (0.47) ALDH1A1CTNNB1WNT3AKMT2AMEN1
SCHEMBL31525615 0.81 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL11790411 0.79 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL28701105 0.79 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL29673203 0.79 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL2775998 0.79 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL3841701 0.79 HDAC1 (0.58) ALDH1A1CYP1A2HPGDL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721942-B1 TETRACYCLIC COMPOUND KYOWA HAKKO KOGYO KK (JP) 2002-06-05 EP disclosed
US-5646283-A IMMUNOSUPPRESSANTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-07-08 US disclosed
EP-0721942-A1 NOVEL TETRACYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-07-17 EP disclosed