SCHEMBL7510044

SCHEMBL7510044

Cc1nc2c(O)cccn2c1C=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 4/20 0.51
GAA P10253 2/20 0.51
LMNA P02545 2/20 0.51
GLA P06280 1/20 0.51
MPI P34949 1/20 0.51
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
BLM P54132 1/20 0.36
ATP4A P20648 2/20 0.36
ATP4B P51164 2/20 0.36
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214205 0.81 ALDH1A1 (0.38) ALDH1A1KDM4EGAAGLAMAPT
SCHEMBL4063787 0.78 ALDH1A1 (0.54) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL9098286 0.77 ALDH1A1 (0.48) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL8816352 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL7016018 0.75 ALDH1A1 (0.56) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL7013857 0.75 KDM4E (0.51) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL9286867 0.74 ALDH1A1 (0.54) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL17028868 0.73 ALDH1A1 (0.50) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL10435571 0.72 ALDH1A1 (0.49) ALDH1A1KDM4EGAALMNAGLA
SCHEMBL5634105 0.72 ATP4A (0.57) ALDH1A1KDM4EGAALMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773946-B1 IMIDAZOPYRIDINE-AZOLIDINONES BYK GULDEN LOMBERG CHEM FAB (DE) 2002-03-27 EP disclosed
EP-0723544-B1 ALKOXY ALKYL CARBAMATES OF IMIDAZO[1,2-a]PYRIDINES BYK GULDEN LOMBERG CHEM FAB (DE) 2001-04-18 EP disclosed
US-6124313-A ACTIVE DRUG FOR TREATING GASTRO-INTESTINAL AILMENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-09-26 US disclosed
EP-0683780-B1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEM FAB (DE) 2000-04-26 EP disclosed
US-5719161-A REACTING AN IMIDAZO(1,2-A)PYRIDINE WITH A PHENYLCARBAMATE; USEFUL IN THE TREATMENT OF GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-02-17 US disclosed
US-5665730-A GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-09-09 US disclosed
EP-0773944-A1 BENZYL-IMIDAZOPYRIDINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1997-05-21 EP disclosed
EP-0773946-A1 IMIDAZOPYRIDINE-AZOLIDINONES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1997-05-21 EP disclosed
EP-0299470-B1 Imidazo[1,2-a]pyridines BYK GULDEN LOMBERG CHEM FAB (DE) 1996-12-04 EP disclosed
EP-0723544-A1 ALKOXY ALKYL CARBAMATES FROM IMIDAZO (1,2-a)PYRIDINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1996-07-31 EP disclosed
WO-1996003405-A1 IMIDAZOPYRIDINE-AZOLIDINONES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-02-08 WO disclosed
EP-0683780-A1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1995-11-29 EP disclosed
WO-1995010518-A1 ALKOXY ALKYL CARBAMATES FROM IMIDAZO (1,2-a)PYRIDINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1995-04-20 WO disclosed
WO-1994018199-A1 IMIDAZOPYRIDINES AND THEIR USE IN TREATING GASTROINTESTINAL DISEASES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-08-18 WO disclosed
US-5112834-A Antisecretory and antiulcer BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1992-05-12 US disclosed
EP-0370056-A1 NEW DIAZOLS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1990-05-30 EP disclosed
WO-1990005136-A1 NEW IMIDAZOPYRIDINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1990-05-17 WO disclosed
EP-0368158-A1 Imidazo pyridines Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1990-05-16 EP disclosed
WO-1989000570-A1 NEW DIAZOLS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1989-01-26 WO disclosed
EP-0299470-A1 Imidazo[1,2-a]pyridines Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1989-01-18 EP disclosed