SCHEMBL7511780

SCHEMBL7511780

O=C(CCCNC(=O)OCc1ccccc1)N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCOC1O

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 1/20 0.51
CAPN1 P07384 1/20 0.48
CTSK P43235 4/20 0.47
CTSB P07858 2/20 0.47
CTSS P25774 2/20 0.47
EPHX2 P34913 1/20 0.47
KLK7 P49862 1/20 0.47
KLK5 Q9Y337 1/20 0.47
HTT P42858 1/20 0.47
CTSL P07711 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515349 0.91 CAPN1 (0.61) CAPN1CTSKCTSSCTSL
SCHEMBL7517799 0.88 BMP1 (0.47) BMP1CAPN1CTSKCTSBCTSS
SCHEMBL8812581 0.87 CTSK (0.60) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL8812573 0.87 CTSK (0.60) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL7511787 0.80 CAPN1 (0.44) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL7512998 0.80 CAPN1 (0.53) BMP1CAPN1CTSKCTSBCTSS
SCHEMBL8810216 0.77 CTSL (0.58) CAPN1CTSKCTSBCTSSKLK7
SCHEMBL8810223 0.77 CTSL (0.58) CAPN1CTSKCTSBCTSSKLK7
SCHEMBL8404288 0.77 CAPN1 (0.68) CAPN1CTSKCTSBCTSSCTSL
SCHEMBL8808396 0.77 CTSK (0.54) CAPN1CTSKCTSBCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed