SCHEMBL7512202

SCHEMBL7512202

CC(C)n1c(=S)[nH]cc(Cc2ccccc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
LGMN Q99538 1/20 0.40
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PNP P00491 1/20 0.38
BRD4 O60885 1/20 0.38
PLK1 P53350 1/20 0.37
HPGD P15428 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7519640 0.88 MEN1 (0.41) L3MBTL1MEN1KMT2AADORA2AADORA1
SCHEMBL18835018 0.80 GFER (0.45) ALDH1A1MEN1KMT2AADORA2AADORA1
SCHEMBL10281157 0.76 ALDH1A1 (0.43) ALDH1A1L3MBTL1KMT2AMAPTPLK1
SCHEMBL27973711 0.73 MEN1 (0.37) ALDH1A1L3MBTL1MEN1KMT2AADORA2A
SCHEMBL8656134 0.71 ALDH1A1 (0.47) ALDH1A1L3MBTL1SMN1; SMN2MAPTPLK1
SCHEMBL7741672 0.68 PLA2G7 (0.41) ALDH1A1MEN1KMT2ALGMNSMN1; SMN2
SCHEMBL4418633 0.68 ALDH1A1 (0.53) ALDH1A1MEN1KMT2ASMN1; SMN2PNP
SCHEMBL17446077 0.67 NPC1 (0.59) ALDH1A1L3MBTL1MEN1KMT2ASMN1; SMN2
SCHEMBL5223001 0.67 KMT2A (0.62) ALDH1A1MEN1KMT2AADORA2AADORA1
SCHEMBL12794269 0.67 PDE3B (0.42) ALDH1A1L3MBTL1KMT2APDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1352637-A Process for preparing MKC-442 TRIANGLE PHARMACEUTICALS INC (US) 2002-06-05 CN disclosed
EP-1169310-A1 PROCESS FOR PREPARING MKC-442 Triangle Pharmaceuticals Inc. (US) 2002-01-09 EP disclosed
EP-1169310-A1 PROCESS FOR PREPARING MKC-442 Triangle Pharmaceuticals Inc. (US) 2002-01-09 EP disclosed
WO-2000061566-A1 PROCESS FOR PREPARING MKC-442 TRIANGLE PHARMACEUTICALS, INC. (US) 2000-10-19 WO disclosed
WO-2000061566-A1 PROCESS FOR PREPARING MKC-442 TRIANGLE PHARMACEUTICALS, INC. (US) 2000-10-19 WO disclosed