SCHEMBL7512877

SCHEMBL7512877

Cc1cccc(CCc2oc(C)nc2C(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.45
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
DAO P14920 2/20 0.40
PIN1 Q13526 1/20 0.40
AKR1C3 P42330 1/20 0.40
CTBP2 P56545 1/20 0.40
GPR84 Q9NQS5 1/20 0.39
SLC7A11 Q9UPY5 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501660 0.88 SORT1 (0.40) ALDH1A1KMT2ASLC7A11NPC1RAB9A
SCHEMBL7508066 0.88 BCL2 (0.40) ALDH1A1KMT2ASLC7A11NPC1
SCHEMBL11741106 0.87 P2RX3 (0.44) ALDH1A1KMT2ADAOSLC7A11NPC1
SCHEMBL7508419 0.87 ALDH1A1 (0.47) ALDH1A1KMT2ATAAR1PIN1NPC1
SCHEMBL7512815 0.78 NR3C2 (0.45) NR3C2ALDH1A1KMT2ATAAR1DAO
SCHEMBL7507225 0.78 NR3C2 (0.45) NR3C2ALDH1A1KMT2ATAAR1DAO
SCHEMBL754250 0.78 EGLN1 (0.42) NR3C2ALDH1A1KMT2A
SCHEMBL11747526 0.76 P2RX3 (0.40) ALDH1A1KMT2ATAAR1RAB9A
SCHEMBL11829444 0.74 CES1 (0.45) ALDH1A1RAB9AL3MBTL1
SCHEMBL11739215 0.73 ALDH1A1 (0.50) ALDH1A1KMT2ANPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042320-B1 NEW COMPOUNDS WHICH ARE P2-PURINOCEPTOR 7-TRANSMEMBRANE (TM) G-PROTEIN COUPLED RECEPTOR ANTAGONISTS ASTRAZENECA UK LTD (GB) 2002-02-13 EP disclosed
US-6218376-B1 FOR TREATING INFLAMMATORY DISEASES ASTRAZENECA UK LIMITED (GB) 2001-04-17 US disclosed
EP-1042320-A1 NEW COMPOUNDS WHICH ARE P2-PURINOCEPTOR 7-TRANSMEMBRANE (TM) G-PROTEIN COUPLED RECEPTOR ANTAGONISTS AstraZeneca UK Limited (GB) 2000-10-11 EP disclosed
WO-1999026944-A1 NEW COMPOUNDS WHICH ARE P2-PURINOCEPTOR 7-TRANSMEMBRANE (TM) G-PROTEIN COUPLED RECEPTOR ANTAGONISTS ASTRAZENEKA UK LIMITED (GB) 1999-06-03 WO disclosed